首页 工具
登录
购物车

搜索结果

Search Results for " vmat2 inhibitor "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T7147 Valbenazine

NBI-98854

Monoamine Transporter Membrane transporter/Ion channel
Valbenazine (NBI-98854) 是一种高度选择性的囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,Ki 为 110-190 nM,用于治疗迟发性运动障碍。
T0719 Tetrabenazine

Xenazine,丁苯那嗪,Ro 1-9569

Others; Dopamine Receptor; Monoamine Transporter GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience; Others
Tetrabenazine (Ro 1-9569) 是 VMAT 抑制剂,用作抗精神病药和治疗各种运动障碍。
T13134 (+)-Tetrabenazine

(+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ

Monoamine Transporter Membrane transporter/Ion channel
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) 是一种可逆的囊泡单胺转运蛋白2 (VMAT-2)抑制剂,对 VMAT2转运的抑制作用是VMAT1的10倍。
T13133 Tetrabenazine Metabolite

(-)-β-Dihydrotetrabenazine,(-)-β-HTBZ

Monoamine Transporter Membrane transporter/Ion channel
Tetrabenazine Metabolite ((-)-β-HTBZ) 是一种囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,是 Tetrabenazine 的一种活性代谢物。Tetrabenazine Metabolite 对 VMAT2 具有高亲和力,其Ki 为13.4 nM。Tetrabenazine Metabolite 常常被用于研究与亨廷顿氏病和其他多动障碍相关的舞蹈病。
T24941 VMAT2-IN-I HCl

VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride

VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.
T79061 VMAT2-IN-2 tosylate

Monoamine Transporter Membrane transporter/Ion channel
VMAT2-IN-2 tosylate,作为VMAT2的有效抑制剂,应用于迟发性运动障碍的研究。
T25750 Lobelane Hydrochloride

Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor.
T22452 Valbenazine tosylate

結苯那嗪,NBI-98854

Monoamine Transporter Membrane transporter/Ion channel
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).

化合物

Valbenazine
Cat.No: T7147
Synonym: NBI-98854
Target: Monoamine Transporter
Tetrabenazine
Cat.No: T0719
Synonym: Xenazine,丁苯那嗪,Ro 1-9569
Target: Others, Dopamine Receptor, Monoamine Transporter
(+)-Tetrabenazine
Cat.No: T13134
Synonym: (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ
Target: Monoamine Transporter
Tetrabenazine Metabolite
Cat.No: T13133
Synonym: (-)-β-Dihydrotetrabenazine,(-)-β-HTBZ
Target: Monoamine Transporter
VMAT2-IN-I HCl
Cat.No: T24941
Synonym: VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride
Target:
VMAT2-IN-2 tosylate
Cat.No: T79061
Synonym:
Target: Monoamine Transporter
Lobelane Hydrochloride
Cat.No: T25750
Synonym:
Target:
Valbenazine tosylate
Cat.No: T22452
Synonym: 結苯那嗪,NBI-98854
Target: Monoamine Transporter
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼