Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7147 |
Valbenazine
NBI-98854 |
Monoamine Transporter | Membrane transporter/Ion channel |
Valbenazine (NBI-98854) 是一种高度选择性的囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,Ki 为 110-190 nM,用于治疗迟发性运动障碍。 | |||
T0719 |
Tetrabenazine
Xenazine,丁苯那嗪,Ro 1-9569 |
Others; Dopamine Receptor; Monoamine Transporter | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience; Others |
Tetrabenazine (Ro 1-9569) 是 VMAT 抑制剂,用作抗精神病药和治疗各种运动障碍。 | |||
T13134 |
(+)-Tetrabenazine
(+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ |
Monoamine Transporter | Membrane transporter/Ion channel |
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) 是一种可逆的囊泡单胺转运蛋白2 (VMAT-2)抑制剂,对 VMAT2转运的抑制作用是VMAT1的10倍。 | |||
T13133 |
Tetrabenazine Metabolite
(-)-β-Dihydrotetrabenazine,(-)-β-HTBZ |
Monoamine Transporter | Membrane transporter/Ion channel |
Tetrabenazine Metabolite ((-)-β-HTBZ) 是一种囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,是 Tetrabenazine 的一种活性代谢物。Tetrabenazine Metabolite 对 VMAT2 具有高亲和力,其Ki 为13.4 nM。Tetrabenazine Metabolite 常常被用于研究与亨廷顿氏病和其他多动障碍相关的舞蹈病。 | |||
T24941 |
VMAT2-IN-I HCl
VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride |
||
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A. | |||
T79061 | VMAT2-IN-2 tosylate | Monoamine Transporter | Membrane transporter/Ion channel |
VMAT2-IN-2 tosylate,作为VMAT2的有效抑制剂,应用于迟发性运动障碍的研究。 | |||
T25750 |
Lobelane Hydrochloride
|
||
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor. | |||
T22452 |
Valbenazine tosylate
結苯那嗪,NBI-98854 |
Monoamine Transporter | Membrane transporter/Ion channel |
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM). |